Copper-Mediated Amidation of Heterocyclic and Aromatic C−H Bonds
| Title: | Copper-Mediated Amidation of Heterocyclic and Aromatic C−H Bonds |
| Author: |
Wang, Qiu; Schreiber, Stuart L.
Note: Order does not necessarily reflect citation order of authors. |
| Citation: | Wang, Qiu, and Stuart L. Schreiber. 2009. Copper-mediated amidation of heterocyclic and aromatic C−H bonds. Organic Letters 11(22): 5178-5180. |
| Full Text & Related Files: |
2776381.pdf (212.5Kb; PDF) 
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| Abstract: | A copper-mediated aerobic coupling reaction enables direct amidation of heterocycles or aromatics having weakly acidic C−H bonds with a variety of nitrogen nucleophiles. These reactions provide efficient access to many biologically important skeletons, including ones with the potential to serve as inhibitors of HMTs. |
| Published Version: | doi:10.1021/ol902079g |
| Other Sources: | http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2776381/pdf/ |
| Terms of Use: | This article is made available under the terms and conditions applicable to Open Access Policy Articles, as set forth at http://nrs.harvard.edu/urn-3:HUL.InstRepos:dash.current.terms-of-use#OAP |
| Citable link to this page: | http://nrs.harvard.edu/urn-3:HUL.InstRepos:4459010 |
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